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Optimization of the Natural Product Calothrixin A to Discover Novel Dual Topoisomerase I and II Inhibitors with Improved Anticancer Activity 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 11, 页码: 8040-8061
作者:  Yang, Xiaohong;  Wang, Zhi-Peng;  Xiang, Sichuan;  Wang, Daoqiang;  Zhao, Yi;  Luo, Dong;  Qiu, Yanfei;  Huang, Chao;  Guo, Jian;  Dai, Yuanwei;  Zhang, Shao-Lin;  He, Yun
收藏  |  浏览/下载:38/0  |  提交时间:2022/08/22
Glutathione-responsive multifunctional nanoparticles based on mannose-modified pillar[5]arene for targeted antibiotic delivery against intracellular methicillin-resistant S. aureus 期刊论文
MATERIALS CHEMISTRY FRONTIERS, 2021, 页码: 8
作者:  Peng, Haibo;  Xie, Beibei;  Cen, Xianfeng;  Dai, Jiaojiao;  Dai, Yuanwei;  Yang, Xiaohong;  He, Yun
收藏  |  浏览/下载:40/0  |  提交时间:2022/08/22
Hollow and Porous Fe3C-NC Nanoballoons Nanozymes for Cancer Cell H2O(2 )Detection 期刊论文
SENSORS AND ACTUATORS B-CHEMICAL, 2021, 卷号: 347, 页码: 7
作者:  Xie, Beibei;  Yang, Xiaohong;  Zhang, Ruixue;  Guo, Jian;  Chen, Zichao;  He, Yun
收藏  |  浏览/下载:168/0  |  提交时间:2021/11/26
Fe  N  C catalysts  Nanozymes  Fluorescent probe  Biosensors  
Synthesis, biological evaluation and structure-activity relationship of novel dichloroacetophenones targeting pyruvate dehydrogenase kinases with potent anticancer activity 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 214, 页码: 16
作者:  Xu, Biao;  Wang, Zhi-Peng;  Liu, Qingwang;  Yang, Xiaohong;  Li, Xuemin;  Huang, Ding;  Qiu, Yanfei;  Tam, Kin Yip;  Zhang, Shao-Lin;  He, Yun
收藏  |  浏览/下载:78/0  |  提交时间:2021/05/17
Pyruvate dehydrogenase kinase  Proliferation  Cancer metabolism  Structure-activity relationship  
Eradicating intracellular MRSA via targeted delivery of lysostaphin and vancomycin with mannose-modified exosomes 期刊论文
JOURNAL OF CONTROLLED RELEASE, 2021, 卷号: 329, 页码: 454-467
作者:  Yang, Xiaohong;  Xie, Beibei;  Peng, Haibo;  Shi, Gongming;  Sreenivas, Banne;  Guo, Jian;  Wang, Chenhui;  He, Yun
收藏  |  浏览/下载:126/0  |  提交时间:2021/05/17
Exosomes  Surface functionalization  Antibiotics  Targeted delivery  Intracellular infection  
Pillar[5]arene-based, dual pH and enzyme responsive supramolecular vesicles for targeted antibiotic delivery against intracellular MRSA 期刊论文
CHEMICAL COMMUNICATIONS, 2020, 卷号: 56, 期号: 58, 页码: 8115-8118
作者:  Peng, Haibo;  Xie, Beibei;  Yang, Xiaohong;  Dai, Jiaojiao;  Wei, Guoxing;  He, Yun
收藏  |  浏览/下载:99/0  |  提交时间:2020/08/24